SCHEMBL2005283

SCHEMBL2005283

O=C(c1ncc(-c2ccncc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGES2 Q9H7Z7 1/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35
TUBA1A Q71U36 1/20 0.35
TUBA1C Q9BQE3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2003933 0.94 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2006671 0.91 PTGES2 (0.40) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2004214 0.91 CCR9 (0.37) KDM4EMEN1KMT2APTGES2MCHR1
SCHEMBL2003600 0.89 LMNA (0.40) ALDH1A1MEN1LMNAPOLBKMT2A
SCHEMBL2002457 0.89 ALOX5 (0.36) ALDH1A1KDM4ELMNAPTGES2MCHR1
SCHEMBL2000914 0.89 FAAH (0.42) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2005131 0.88 FAAH (0.41) KDM4EMEN1KMT2APTGES2CYP1A2
SCHEMBL2008226 0.88 ALDH1A1 (0.41) ALDH1A1KDM4EMEN1USP2LMNA
SCHEMBL2001282 0.88 FAAH (0.42)
SCHEMBL2002560 0.87 MAPT (0.40) MEN1KMT2APTGES2CYP3A4CCR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed