SCHEMBL2005131

SCHEMBL2005131

Cc1ccc2c(c1)c(C(=O)c1ncc(-c3ccncc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
PTGES2 Q9H7Z7 8/20 0.36
ALOX5 P09917 1/20 0.36
ALOX5AP P20292 1/20 0.36
CCR9 P51686 1/20 0.35
MAPT P10636 2/20 0.34
CYP2C9 P11712 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004214 0.93 CCR9 (0.37) FAAHMEN1KMT2APTGES2ALOX5
SCHEMBL2001077 0.93 PTGES2 (0.41) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2005859 0.91 PTGES2 (0.44) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2002457 0.91 ALOX5 (0.36) PTGES2ALOX5ALOX5APCCR9MAPT
SCHEMBL2002947 0.91 CYP3A4 (0.35) FAAHMAPTCYP2C9CYP3A4PTGDR2
SCHEMBL1998915 0.90 LMNA (0.42) FAAHMEN1KMT2AALOX5ALOX5AP
SCHEMBL2006590 0.90 FAAH (0.40) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2001753 0.89 FAAH (0.44) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2001878 0.89 ALOX5AP (0.42) KMT2AALOX5ALOX5APMAPTCYP2C9
SCHEMBL2005283 0.88 ALDH1A1 (0.38) MEN1KMT2APTGES2CCR9CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed