SCHEMBL20053804

SCHEMBL20053804

CSc1ccc(Cl)cc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
TP53 P04637 1/20 0.57
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
TSHR P16473 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
CASP1 P29466 1/20 0.52
KDM4E B2RXH2 2/20 0.50
HSD17B10 Q99714 1/20 0.50
MYC P01106 2/20 0.49
NR4A1 P22736 1/20 0.49
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
F7 P08709 1/20 0.43
F3 P13726 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7492153 0.85 HTT (0.44) ALDH1A1TP53CA1CA2SMN1; SMN2
SCHEMBL10334495 0.85 SMN1; SMN2 (0.57) ALDH1A1TP53CA1CA2TSHR
SCHEMBL4437995 0.84 ALDH1A1 (0.61) ALDH1A1TP53CA1CA2TSHR
SCHEMBL823686 0.84 ALDH1A1 (0.61) ALDH1A1TP53CA1CA2TSHR
SCHEMBL11765343 0.83 ALDH1A1 (0.47) ALDH1A1TP53CA1CA2TSHR
SCHEMBL12505458 0.83 KDM4E (0.54) ALDH1A1TP53CA1CA2SMN1; SMN2
SCHEMBL1262469 0.80 ABL1 (0.56) ALDH1A1TSHRSMN1; SMN2KDM4EGAA
SCHEMBL31620799 0.80 ABL1 (0.56) ALDH1A1TSHRSMN1; SMN2KDM4EGAA
SCHEMBL12164877 0.80 ADRA1D (0.43) ALDH1A1TP53CA1CA2SMN1; SMN2
SCHEMBL16954098 0.80 CCR2 (0.40) ALDH1A1TP53CA1CA2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10570148-B2 N-alkyl-2-phenoxyethanamines, their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2020-02-25 US disclosed
US-20180222919-A1 N-ALKYL-2-PHENOXYETHANAMINES, THEIR PREPARATION AND USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-08-09 US disclosed
US-9944644-B2 Octahydropyrrolopyrroles their preparation and use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10570148-B2 N-alkyl-2-phenoxyethanamines, their preparation and use HRH3, CBR3, KCNH3 ALDH1A1 2874/4885TP53 3119/4885CA1 2151/4885
US-20180222919-A1 N-ALKYL-2-PHENOXYETHANAMINES, THEIR PREPARATION AND USE HRH3, CBR3, KCNH3 ALDH1A1 2874/4885TP53 3119/4885CA1 2151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.