SCHEMBL2005776

SCHEMBL2005776

COc1ccc2c(c1)c(C(=O)c1nnc(-c3ccncn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 4/20 0.37
PTGS2 P35354 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
GSK3B P49841 1/20 0.34
PDE4B Q07343 1/20 0.33
PDE11A Q9HCR9 1/20 0.33
MAPT P10636 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
MEN1 O00255 1/20 0.33
RGS12 O14924 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
GNAI1 P63096 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004327 0.94 F2RL3 (0.34) PLA2G2APDE4BPDE11AMAPTCYP3A4
SCHEMBL2003824 0.93 LMNA (0.33) GSK3BPDE4BPDE11AMAPTCYP1A2
SCHEMBL2004842 0.91 FAAH (0.33) PTGDR2PDE4BPDE11AMAPTALDH1A1
SCHEMBL2007916 0.91 LMNA (0.41) PLA2G2APTGS2MAPTCYP1A2CYP3A4
SCHEMBL2003372 0.91 PLA2G2A (0.38) PLA2G2APTGS2PTGDR2GSK3BMAPT
SCHEMBL2002081 0.91 L3MBTL1 (0.35) PDE4BPDE11AMAPTALDH1A1LMNA
SCHEMBL2005382 0.90 PLA2G2A (0.38) PLA2G2APTGDR2GSK3BMAPTCYP1A2
SCHEMBL2007059 0.90 MAPK1 (0.41) PLA2G2APTGS2PTGDR2GSK3BPDE4B
SCHEMBL2008174 0.90 PLA2G2A (0.42) PLA2G2APTGDR2MAPTCYP1A2CYP3A4
SCHEMBL2010346 0.89 PLA2G2A (0.37) PLA2G2APTGS2PTGDR2GSK3BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed