SCHEMBL2003372

SCHEMBL2003372

COc1ccc2c(c1)c(C(=O)c1nnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 6/20 0.38
OPRK1 P41145 1/20 0.37
PTGS2 P35354 1/20 0.36
F2RL3 Q96RI0 2/20 0.35
ACHE P22303 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
MAPT P10636 1/20 0.34
ALOX5AP P20292 1/20 0.34
GSK3B P49841 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2004340 0.94 F2RL3 (0.37) OPRK1F2RL3MAPTALOX5APKDM4E
SCHEMBL2004659 0.93 KDM4E (0.37) OPRK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4544118 0.92 OPRK1 (0.38) PLA2G2AOPRK1ACHECYP1A2CYP3A4
SCHEMBL2001936 0.91 OPRK1 (0.36) OPRK1CYP1A2CYP2D6CYP2C9MAPT
SCHEMBL2004726 0.91 OPRK1 (0.42) PLA2G2AOPRK1PTGS2ACHECYP1A2
SCHEMBL2005776 0.91 PLA2G2A (0.37) PLA2G2APTGS2F2RL3CYP1A2CYP3A4
SCHEMBL2008404 0.90 L3MBTL1 (0.39) OPRK1CYP1A2CYP2D6CYP2C9MAPT
SCHEMBL1999938 0.90 PLA2G2A (0.39) PLA2G2AACHEPTGDR2MAPTGSK3B
SCHEMBL2003477 0.90 LMNA (0.40) OPRK1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2003008 0.90 PLA2G2A (0.40) PLA2G2APTGS2F2RL3CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed