SCHEMBL20057789

SCHEMBL20057789

Cc1c(-c2ccccc2)ncn1-c1ccc(C=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
SMN1; SMN2 Q16637 2/20 0.45
GPR119 Q8TDV5 1/20 0.44
FAAH O00519 2/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GRM1 Q13255 2/20 0.38
CYP2A6 P11509 1/20 0.38
PTGS2 P35354 2/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
FGFR1 P11362 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15507102 0.81 GPR119 (0.53) ALDH1A1SMN1; SMN2GPR119FAAHMEN1
SCHEMBL29205308 0.77 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2KDM4ECYP2A6PTGS2
SCHEMBL28760303 0.76 MAPK9 (0.47) ALDH1A1SMN1; SMN2GPR119FAAH
SCHEMBL23884857 0.74 ALDH1A1 (0.62) ALDH1A1MEN1KMT2AKDM4ECYP2A6
SCHEMBL11442828 0.73 KDM4E (0.41) ALDH1A1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL27662257 0.72 L3MBTL1 (0.47) ALDH1A1SMN1; SMN2GPR119FAAHLMNA
SCHEMBL2568999 0.68 FGFR1 (0.72) ALDH1A1KDM4EHTTFGFR1
SCHEMBL29512158 0.68 FGFR1 (0.72) ALDH1A1KDM4EHTTFGFR1
SCHEMBL24311359 0.68 HTT (0.49) ALDH1A1SMN1; SMN2MITFLMNAHTT
SCHEMBL24528609 0.68 XDH (0.44) ALDH1A1GRM1PTGS2FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892888-B1 N-CYCLOPROPYL-N-PIPERIDINYL-AMIDES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed