SCHEMBL20060147

SCHEMBL20060147

CN/C(=C1\C(=N)CCCC1=O)c1cccc(C)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
HPD P32754 7/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060183 0.87 NPC1 (0.35) HPD
SCHEMBL20060194 0.83 ALDH1A1 (0.37) HPD
SCHEMBL20060133 0.78 HPD (0.34) P2RX7HPD
SCHEMBL20060137 0.77 P2RX7 (0.36) P2RX7TAS1R3TAS1R1TAS1R2
SCHEMBL20060196 0.77 CTSD (0.39) HPD
SCHEMBL20059994 0.77 NPC1 (0.36)
SCHEMBL20060177 0.74 HPD (0.36) HPD
SCHEMBL20059914 0.74 HPD (0.40) P2RX7HPD
SCHEMBL20059923 0.74 HPD (0.40) P2RX7HPD
SCHEMBL20060130 0.72 GRIN1 (0.40) P2RX7TAS1R3TAS1R1TAS1R2HPD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed