SCHEMBL20060177

SCHEMBL20060177

CN/C(=C1\C(=N)CCCC1=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HPD P32754 5/20 0.36
MAPT P10636 1/20 0.36
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060183 0.81 NPC1 (0.35) HPDMAPTNPC1ALDH1A1POLB
SCHEMBL20060194 0.80 ALDH1A1 (0.37) HPDMAPTNPC1ALDH1A1POLB
SCHEMBL20060196 0.79 CTSD (0.39) HPDMAPTNPC1ALDH1A1RAB9A
SCHEMBL20060138 0.77 RAB9A (0.38) MAPTNPC1ALDH1A1POLBRAB9A
SCHEMBL18235403 0.77 HPD (0.38) HPDNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL20060147 0.74 P2RX7 (0.38) HPD
SCHEMBL20060173 0.73 KDM4E (0.35) MAPTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL20060139 0.73 CMA1 (0.39) HPDMAPTNPC1ALDH1A1TSHR
SCHEMBL20059994 0.73 NPC1 (0.36) MAPTNPC1ALDH1A1POLBRAB9A
SCHEMBL20060195 0.72 MEN1 (0.40) ALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed