SCHEMBL20060195

SCHEMBL20060195

CCC(/C(NC)=C1/C(=N)CCCC1=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 2/20 0.37
KCNQ2 O43526 4/20 0.37
KCNQ3 O43525 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
KCNE1 P15382 1/20 0.37
KCNQ1 P51787 1/20 0.37
KCNQ4 P56696 1/20 0.37
POLB P06746 1/20 0.36
LMNA P02545 2/20 0.36
HSD17B10 Q99714 1/20 0.36
CRHBP P24387 2/20 0.36
CRHR2 Q13324 2/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20060143 0.81 ALDH1A1 (0.36) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL20060030 0.76 KCNQ2 (0.37) MEN1KMT2AALDH1A1KCNQ2POLB
SCHEMBL20060177 0.72 HPD (0.36) ALDH1A1POLBSMN1; SMN2
SCHEMBL20060139 0.70 CMA1 (0.39) ALDH1A1HTT
SCHEMBL20060020 0.68 MEN1 (0.30) MEN1KMT2AALDH1A1
SCHEMBL20060183 0.67 NPC1 (0.35) MEN1KMT2AALDH1A1CYP3A4CYP2C9
SCHEMBL20060136 0.66 MEN1 (0.37) MEN1KMT2AALDH1A1
SCHEMBL2049579 0.66 ALDH1A1 (0.66) MEN1KMT2AALDH1A1KCNQ2CYP1A2
SCHEMBL20059919 0.66 MEN1 (0.35) MEN1KMT2AALDH1A1
SCHEMBL10192825 0.66 LMNA (0.47) MEN1KMT2AALDH1A1KCNQ2KCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed