SCHEMBL2006387

SCHEMBL2006387

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
MCL1 Q07820 1/20 0.39
MEN1 O00255 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
PTGES2 Q9H7Z7 6/20 0.38
ALOX5AP P20292 5/20 0.38
PTGS1 P23219 1/20 0.38
PTGES O14684 1/20 0.37
CYP3A4 P08684 1/20 0.36
ALOX5 P09917 1/20 0.36
CYP2C9 P11712 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009144 0.93 CYP3A4 (0.38) MCL1MEN1KMT2APTGES2ALOX5AP
SCHEMBL2002269 0.92 LMNA (0.35) FAAHMCL1MEN1HTTKMT2A
SCHEMBL2007516 0.91 S1PR3 (0.38) MCL1MEN1KMT2APTGES2ALOX5AP
SCHEMBL2003713 0.91 MCL1 (0.39) MCL1MEN1KMT2APTGES2CYP3A4
SCHEMBL2002780 0.90 ACHE (0.44) MEN1KMT2AALOX5APCYP3A4ALOX5
SCHEMBL2007874 0.89 FAAH (0.41) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2010143 0.89 PTGES2 (0.42) FAAHMEN1HTTKMT2APTGES2
SCHEMBL2006280 0.89 FAAH (0.44) FAAHMCL1MEN1HTTKMT2A
SCHEMBL1999807 0.89 ALOX5AP (0.42) ALOX5APPTGS1CYP3A4ALOX5CYP2C9
SCHEMBL2002574 0.89 FAAH (0.42) FAAHMCL1MEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed