SCHEMBL2009144

SCHEMBL2009144

O=C(c1cnc(-c2ccccn2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2)c2ccc(Cl)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
ALOX12 P18054 1/20 0.38
PPARG P37231 1/20 0.38
RECQL P46063 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
ALOX5AP P20292 4/20 0.36
PTGES2 Q9H7Z7 3/20 0.36
ALOX5 P09917 1/20 0.36
CYP2C9 P11712 1/20 0.36
MCL1 Q07820 1/20 0.36
PTGES O14684 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2007516 0.94 S1PR3 (0.38) CYP3A4MEN1MAPTKMT2AALOX5AP
SCHEMBL2003713 0.94 MCL1 (0.39) CYP3A4MEN1KMT2APTGES2CYP2C9
SCHEMBL2006387 0.93 FAAH (0.41) CYP3A4HSD17B10MEN1KMT2AALOX5AP
SCHEMBL2002525 0.93 LMNA (0.38) CYP3A4MEN1MAPTTSHRALOX12
SCHEMBL2002780 0.91 ACHE (0.44) CYP3A4MEN1MAPTTSHRKMT2A
SCHEMBL1999807 0.90 ALOX5AP (0.42) CYP3A4ALOX5APALOX5CYP2C9
SCHEMBL2006787 0.89 PTGES2 (0.36) CYP3A4HSD17B10MEN1MAPTALOX15
SCHEMBL2003741 0.88 MAPT (0.41) CYP3A4HSD17B10MEN1MAPTALOX15
SCHEMBL2001338 0.88 LMNA (0.40) CYP3A4MEN1MAPTTSHRALOX12
SCHEMBL2007882 0.88 HSD17B10 (0.40) CYP3A4HSD17B10MEN1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed