SCHEMBL2002269

SCHEMBL2002269

Cc1ccc2c(c1)c(C(=O)c1cnc(-c3ccccn3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
FAAH O00519 1/20 0.35
MCL1 Q07820 1/20 0.35
OPRK1 P41145 4/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALOX5AP P20292 1/20 0.34
PTGS1 P23219 1/20 0.34
NPSR1 Q6W5P4 3/20 0.34
TSHR P16473 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP3A4 P08684 1/20 0.34
PMP22 Q01453 1/20 0.34
HIF1A Q16665 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002525 0.95 LMNA (0.38) LMNAALDH1A1MAPTALOX12OPRK1
SCHEMBL2006387 0.92 FAAH (0.41) ALDH1A1FAAHMCL1ALOX5APPTGS1
SCHEMBL2001338 0.92 LMNA (0.40) LMNAALDH1A1MAPTALOX12OPRK1
SCHEMBL1999915 0.92 L3MBTL1 (0.39) LMNAALDH1A1MAPTALOX12OPRK1
SCHEMBL2006197 0.91 ACHE (0.39) LMNAALDH1A1MAPTOPRK1ALOX5AP
SCHEMBL2001446 0.90 FAAH (0.35) LMNAALDH1A1MAPTALOX12FAAH
SCHEMBL2002629 0.90 PPARG (0.39) LMNAALDH1A1MAPTALOX12FAAH
SCHEMBL2008873 0.90 LMNA (0.38) LMNAALDH1A1MAPTALOX12FAAH
SCHEMBL2002746 0.90 F2RL3 (0.37) LMNAALDH1A1MAPTALOX12SMN1; SMN2
SCHEMBL2001936 0.88 OPRK1 (0.36) LMNAALDH1A1MAPTALOX12FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed