SCHEMBL20064089

SCHEMBL20064089

CC(C)C(=O)Nc1nc2[nH]cc(I)c2c(=O)[nH]1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.37
KDM4E B2RXH2 4/20 0.36
PAX3 P23760 1/20 0.36
FOXO1 Q12778 1/20 0.36
TSHR P16473 1/20 0.35
GDA Q9Y2T3 1/20 0.35
ADORA3 P0DMS8 2/20 0.34
ADORA2A P29274 1/20 0.32
TP53 P04637 2/20 0.32
MDM4 O15151 1/20 0.32
CHEK1 O14757 1/20 0.32
ALDH1A1 P00352 2/20 0.32
RAF1 P04049 1/20 0.32
BRAF P15056 1/20 0.32
TYMS P04818 1/20 0.32
LMNA P02545 1/20 0.31
HSD17B10 Q99714 1/20 0.31
XIAP P98170 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22639183 0.73 TSHR (0.42) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL442818 0.72 NOS1 (0.45) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL20869901 0.71 TYMS (0.41) TYMS
SCHEMBL22036469 0.69 ALDH1A1 (0.43) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL735411 0.69 GDA (0.72) GDA
SCHEMBL15061831 0.68 TYMS (0.48) KDM4ECHEK1ALDH1A1TYMSLMNA
SCHEMBL18490337 0.68 NOS1 (0.41) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL8886595 0.66 NOS1 (0.38) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL4337068 0.66 PAX3 (0.39) NOS1KDM4EPAX3FOXO1TSHR
SCHEMBL3797825 0.65 SMN1; SMN2 (0.47) KDM4EGDAADORA3ADORA2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018071531-A1 HPPK INHIBITORS USEFUL AS ANTIBACTERIAL AGENTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2018-04-19 WO disclosed