SCHEMBL2007374

SCHEMBL2007374

COc1ccc(F)cc1-c1ccc(C(C)NS(=O)(=O)c2cn(C)nc2C(F)(F)F)c(F)c1

nearest known ligand 0.79

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 6/20 0.79
PGR P06401 4/20 0.79
SGK1 O00141 1/20 0.38
APLNR P35414 2/20 0.37
BRD4 O60885 2/20 0.36
S1PR1 P21453 1/20 0.36
PIK3C3 Q8NEB9 2/20 0.36
FEN1 P39748 3/20 0.36
ALOX5AP P20292 2/20 0.35
CASR P41180 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008107 0.89 NR3C1 (1.00) NR3C1PGRSGK1APLNRBRD4
SCHEMBL2002007 0.79 NR3C1 (0.82) NR3C1PGRSGK1PIK3C3CASR
SCHEMBL2006541 0.77 NR3C1 (0.62) NR3C1PGRSGK1APLNRS1PR1
SCHEMBL2006930 0.77 NR3C1 (0.78) NR3C1PGRS1PR1CASR
SCHEMBL2008089 0.75 NR3C1 (0.79) NR3C1PGRSGK1S1PR1PIK3C3
SCHEMBL2004236 0.73 NR3C1 (0.59) NR3C1PGRBRD4
SCHEMBL2008086 0.69 NR3C1 (0.78) NR3C1PGRSGK1S1PR1PIK3C3
SCHEMBL5237877 0.68 LRRK2 (0.49) NR3C1PGR
SCHEMBL2004688 0.68 ALDH1A1 (0.47) NR3C1PGRS1PR1
SCHEMBL17806608 0.67 PRMT5 (0.45) NR3C1PGRBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960365-B2 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2011-06-14 US disclosed