SCHEMBL2008103

SCHEMBL2008103

CC(NS(=O)(=O)c1ccc(F)c(F)c1)c1ccc(-c2cc(F)cnc2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.40
PGR P06401 3/20 0.40
PTGS2 P35354 5/20 0.39
ALOX5AP P20292 2/20 0.38
FEN1 P39748 1/20 0.38
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 2/20 0.38
CNR1 P21554 3/20 0.37
CNR2 P34972 2/20 0.37
PTGS1 P23219 2/20 0.37
SLC1A3 P43003 1/20 0.37
SLC1A2 P43004 1/20 0.37
SLC1A1 P43005 1/20 0.37
GRM5 P41594 1/20 0.36
EGFR P00533 1/20 0.35
PIK3CA P42336 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2008102 1.00 NR3C1 (0.40) NR3C1PGRPTGS2ALOX5APFEN1
SCHEMBL2005610 0.77 NR3C1 (0.62) NR3C1PGRPTGS2PTGS1ALDH1A1
SCHEMBL2005613 0.77 NR3C1 (0.62) NR3C1PGRPTGS2PTGS1ALDH1A1
SCHEMBL2004275 0.77 NR3C1 (0.51) NR3C1PGRPTGS2CNR1CNR2
SCHEMBL2002894 0.71 ADRB2 (0.42) CNR1EGFR
SCHEMBL2003919 0.71 ADRB2 (0.42) CNR1EGFR
SCHEMBL25705347 0.71 CNR2 (0.44) S1PR1CNR1CNR2
SCHEMBL2406521 0.69 SLC1A3 (0.47) SLC1A3SLC1A2SLC1A1ALDH1A1
SCHEMBL25705360 0.67 GPR55 (0.50) NR3C1PGRPTGS2CNR1PTGS1
SCHEMBL2002174 0.65 NR3C2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960365-B2 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2011-06-14 US disclosed
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2007-06-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor NR3C1, NR3C2, MC2R NR3C1 1/4885PGR 131/4885PTGS2 2428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.