SCHEMBL20085403

SCHEMBL20085403

C=C/C=C(C)\C=C(/C)Cc1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.41
ALDH1A1 P00352 3/20 0.37
RIPK1 Q13546 1/20 0.36
IDO1 P14902 2/20 0.36
CXCL8 P10145 1/20 0.36
LMNA P02545 3/20 0.35
RAB9A P51151 2/20 0.35
MAPK1 P28482 2/20 0.35
NPC1 O15118 1/20 0.35
CASP3 P42574 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
GLS O94925 2/20 0.34
SIGMAR1 Q99720 1/20 0.33
MAOB P27338 1/20 0.33
ELOVL1 Q9BW60 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15066239 0.76 TAAR1 (0.47) TAAR1ALDH1A1RIPK1IDO1CXCL8
SCHEMBL20055723 0.72 TAAR1 (0.34) TAAR1ALDH1A1RIPK1IDO1LMNA
SCHEMBL21886143 0.71 TAAR1 (0.47) TAAR1ALDH1A1RIPK1IDO1LMNA
SCHEMBL172686 0.70 TAAR1 (0.45) TAAR1ALDH1A1RIPK1IDO1LMNA
SCHEMBL13782802 0.70 CES2 (0.36) ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL435759 0.69 TAAR1 (0.48) TAAR1ALDH1A1RIPK1IDO1LMNA
SCHEMBL26375984 0.68 TAAR1 (0.40) TAAR1ALDH1A1IDO1LMNARAB9A
SCHEMBL125583 0.66 ALDH1A1 (0.49) TAAR1ALDH1A1RIPK1IDO1CXCL8
SCHEMBL2206253 0.65 ALDH1A1 (0.48) TAAR1ALDH1A1RIPK1CXCL8LMNA
SCHEMBL29533621 0.64 CXCL8 (0.65) TAAR1ALDH1A1CXCL8LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312172-B1 AMINOPYRAZOLE DERIVATIVES USEFUL AS SRC KINASE INHIBITORS CHUGAI PHARMACEUTICAL CO LTD (JP) 2020-05-06 EP disclosed
EP-3312172-A1 AMINOPYRAZOLE DERIVATIVES Chugai Seiyaku Kabushiki Kaisha (JP) 2018-04-25 EP disclosed