SCHEMBL20094572

SCHEMBL20094572

CC(=O)Nc1c[nH]c(C(=O)NC(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
DAO P14920 5/20 0.40
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
ALOX15 P16050 1/20 0.38
LMNA P02545 1/20 0.38
RORC P51449 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CREBBP Q92793 1/20 0.37
PKM P14618 1/20 0.36
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20094779 0.86 KMT2A (0.45) DAOADORA3ADORA2AADORA2BADORA1
SCHEMBL15318252 0.78 BAZ2B (0.50) GAALMNAALDH1A1TDP1ERCC1
SCHEMBL15318227 0.78 HSD17B10 (0.45) GAADAOLMNAALDH1A1TDP1
SCHEMBL20094767 0.77 DAO (0.49) GAADAOALOX15LMNAALDH1A1
SCHEMBL161465 0.76 ADORA3 (0.43) GAAADORA3ADORA2AADORA2BADORA1
SCHEMBL20094517 0.75 MAPT (0.49) DAOALOX15ALDH1A1PKMSMN1; SMN2
SCHEMBL24740414 0.75 GRN (0.56) GAAADORA3ADORA2AADORA2BADORA1
SCHEMBL20094573 0.73 MMP13 (0.56) ALOX15LMNARORCALDH1A1TDP1
SCHEMBL21180777 0.72 SMN1; SMN2 (0.41) GAAADORA3ADORA2AADORA2BADORA1
SCHEMBL20094768 0.70 KMT2A (0.39) GAADAOLMNAALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018075842-A1 CONDENSED BENZODIAZEPINE DERIVATIVES AND CONJUGATES MADE THEREFROM BRISTOL-MYERS SQUIBB COMPANY (US) 2018-04-26 WO disclosed