SCHEMBL2009502

SCHEMBL2009502

COc1ccc2c(c1)c(C(=O)c1cnc(-c3ccncc3)o1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 5/20 0.38
ALOX5 P09917 1/20 0.38
ALOX5AP P20292 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
RGS12 O14924 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
GNAI1 P63096 1/20 0.37
PMP22 Q01453 1/20 0.37
KMT2A Q03164 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006586 0.93 ALOX5AP (0.39) ALOX5ALOX5APCYP3A4CYP2C9MAPT
SCHEMBL2006531 0.93 PLA2G2A (0.41) PLA2G2AALOX5APCYP1A2CYP3A4CYP2C9
SCHEMBL2001177 0.92 ALOX5AP (0.43) PLA2G2AALOX5ALOX5APCYP1A2CYP3A4
SCHEMBL2004748 0.92 CYP3A4 (0.37) ALOX5ALOX5APCYP1A2CYP3A4CYP2C9
SCHEMBL2010168 0.92 ALOX5AP (0.38) PLA2G2AALOX5ALOX5APCYP1A2CYP3A4
SCHEMBL2006911 0.91 PLA2G2A (0.37) PLA2G2AALOX5ALOX5APCYP1A2CYP3A4
SCHEMBL2008195 0.90 FAAH (0.36) ALOX5ALOX5APCYP3A4CYP2C9MAPT
SCHEMBL2003542 0.90 MAPT (0.39) PLA2G2AALOX5ALOX5APCYP1A2CYP3A4
SCHEMBL2002564 0.89 L3MBTL1 (0.36) ALOX5ALOX5APCYP1A2CYP3A4CYP2C9
SCHEMBL2004143 0.89 LMNA (0.40) CYP1A2CYP3A4CYP2C9MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed