SCHEMBL2004748

SCHEMBL2004748

O=C(c1cnc(-c2ccncc2)o1)c1c(C(F)(F)F)n(Cc2ccc(Cl)cc2Cl)c2ccc(Cl)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
LMNA P02545 2/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
CASP1 P29466 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
PMP22 Q01453 1/20 0.33
HIF1A Q16665 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALOX5 P09917 1/20 0.33
ALOX5AP P20292 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2002564 0.95 L3MBTL1 (0.36) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2008195 0.94 FAAH (0.36) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2004143 0.94 LMNA (0.40) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2009968 0.92 MAPT (0.39) CYP3A4CYP2C9LMNATSHRKMT2A
SCHEMBL2009502 0.92 PLA2G2A (0.38) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2003925 0.92 ALOX5 (0.39) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2006586 0.92 ALOX5AP (0.39) CYP3A4CYP2C9LMNAMAPTALOX5
SCHEMBL2001072 0.91 PTGES2 (0.38) CYP3A4CYP2C9LMNATSHRALDH1A1
SCHEMBL2004795 0.90 MAPT (0.34) CYP3A4CYP2C9LMNATSHRMAPK1
SCHEMBL2004625 0.89 CYP2C9 (0.40) CYP3A4CYP2C9LMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed