SCHEMBL2009722

SCHEMBL2009722

O=C(N[C@@H]1CON(C2CSC2)C1=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
PKM P14618 1/20 0.47
CASP1 P29466 1/20 0.45
CASP8 Q14790 1/20 0.45
SRC P12931 4/20 0.42
KDM4E B2RXH2 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
RIPK1 Q13546 1/20 0.39
HTT P42858 1/20 0.39
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2009724 1.00 ALDH1A1 (0.47) ALDH1A1PKMCASP1CASP8SRC
SCHEMBL2033656 0.74 RIPK1 (0.45) ALDH1A1PKMDDB1CRBNRIPK1
SCHEMBL5903467 0.70 CASP1 (0.67) ALDH1A1PKMCASP1CASP8SRC
SCHEMBL15688484 0.69 NPC1 (0.56) ALDH1A1PKMKDM4E
SCHEMBL11840921 0.69 ALDH1A1 (0.68) ALDH1A1PKMCASP1CASP8SRC
SCHEMBL1936056 0.68 ALDH1A1 (0.71) ALDH1A1PKMKDM4EDDB1CRBN
SCHEMBL1456877 0.64 MEN1 (0.58) ALDH1A1PKMKDM4ENFKB1NFKB2
SCHEMBL1456878 0.64 MEN1 (0.58) ALDH1A1PKMKDM4ENFKB1NFKB2
SCHEMBL1907404 0.64 MEN1 (0.58) ALDH1A1PKMKDM4ENFKB1NFKB2
SCHEMBL10713076 0.64 NAMPT (0.55) ALDH1A1DDB1CRBNHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2507230-A1 INSECTICIDAL COMPOUNDS BASED ON ISOXAZOLINE DERIVATIVES Syngenta Participations AG (CH) 2012-10-10 EP disclosed
WO-2011067272-A1 INSECTICIDAL COMPOUNDS BASED ON ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed