SCHEMBL20103463

SCHEMBL20103463

S=C(Nc1ccc(OCc2nc3ccccc3[nH]2)cc1)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.59
SMN1; SMN2 Q16637 8/20 0.59
NPC1 O15118 7/20 0.59
POLB P06746 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
TP53 P04637 2/20 0.54
TSHR P16473 1/20 0.54
LMNA P02545 3/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 2/20 0.53
MEN1 O00255 1/20 0.53
GAA P10253 1/20 0.53
MAPK1 P28482 1/20 0.53
ALDH1A1 P00352 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
KDM4E B2RXH2 1/20 0.52
ALOX5 P09917 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103496 0.90 ALOX5 (0.63) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL20103483 0.89 ALOX5 (0.53) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL20103473 0.79 ALOX5 (0.67) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL6524094 0.78 MAPT (0.53) POLBTDP1TP53LMNAKMT2A
SCHEMBL20103462 0.76 NPC1 (0.47) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL14642400 0.76 TP53 (0.62) TP53LMNAKMT2AHTTMEN1
SCHEMBL20103615 0.76 NPC1 (0.56) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL2245506 0.75 RAB9A (1.00) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL2241896 0.72 RAB9A (1.00) RAB9ASMN1; SMN2NPC1POLBTDP1
SCHEMBL13679571 0.72 TP53 (0.53) RAB9ASMN1; SMN2NPC1TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed