SCHEMBL20103473

SCHEMBL20103473

Cc1cc(OCc2nc3ccccc3[nH]2)ccc1NC(=O)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.67
EPHX2 P34913 7/20 0.67
ALOX5AP P20292 1/20 0.67
NTRK1 P04629 5/20 0.57
NTRK2 Q16620 3/20 0.57
LMNA P02545 2/20 0.52
GAA P10253 2/20 0.52
MAPT P10636 2/20 0.52
SMN1; SMN2 Q16637 4/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
TP53 P04637 2/20 0.48
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103483 0.89 ALOX5 (0.53) ALOX5EPHX2ALOX5APNTRK1NTRK2
SCHEMBL20103496 0.89 ALOX5 (0.63) ALOX5EPHX2NTRK1NTRK2LMNA
SCHEMBL20103574 0.80 ALOX5 (0.67) ALOX5EPHX2ALOX5APMAPTSMN1; SMN2
SCHEMBL20103602 0.80 EPHX2 (1.00) ALOX5EPHX2ALOX5AP
SCHEMBL20103463 0.79 RAB9A (0.59) ALOX5EPHX2LMNAGAAMAPT
SCHEMBL20103550 0.77 NPC1 (0.64) LMNAGAASMN1; SMN2NPC1RAB9A
SCHEMBL6524094 0.77 MAPT (0.53) NTRK1NTRK2LMNAMAPTTP53
SCHEMBL13945712 0.71 EPHX2 (0.54) ALOX5EPHX2ALOX5APLMNAGAA
SCHEMBL14332504 0.69 TP53 (0.82) LMNAMAPTSMN1; SMN2TP53MEN1
SCHEMBL20103594 0.69 EPHX2 (0.64) ALOX5EPHX2ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed