SCHEMBL20103496

SCHEMBL20103496

O=C(Nc1ccc(OCc2nc3ccccc3[nH]2)cc1)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.63
EPHX2 P34913 1/20 0.63
NTRK1 P04629 6/20 0.59
NTRK2 Q16620 4/20 0.59
NPC1 O15118 7/20 0.59
RAB9A P51151 7/20 0.59
SMN1; SMN2 Q16637 6/20 0.59
POLB P06746 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
ALDH1A1 P00352 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C19 P33261 1/20 0.57
TP53 P04637 2/20 0.54
TSHR P16473 1/20 0.54
LMNA P02545 2/20 0.53
HTT P42858 2/20 0.53
PKM P14618 1/20 0.53
KMT2A Q03164 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20103463 0.90 RAB9A (0.59) ALOX5EPHX2NPC1RAB9ASMN1; SMN2
SCHEMBL20103473 0.89 ALOX5 (0.67) ALOX5EPHX2NTRK1NTRK2NPC1
SCHEMBL6524094 0.83 MAPT (0.53) NTRK1NTRK2POLBTDP1ALDH1A1
SCHEMBL20103483 0.79 ALOX5 (0.53) ALOX5EPHX2NTRK1NTRK2NPC1
SCHEMBL20103600 0.77 EPHX2 (0.63) ALOX5EPHX2NPC1RAB9ATP53
SCHEMBL2245506 0.75 RAB9A (1.00) NPC1RAB9ASMN1; SMN2POLBTDP1
SCHEMBL14615298 0.73 MAPT (0.72) TP53LMNAHTTKMT2AMEN1
SCHEMBL29518652 0.73 NPC1 (0.54) NPC1RAB9ASMN1; SMN2TDP1LMNA
SCHEMBL28372308 0.73 NPC1 (0.54) NPC1RAB9ASMN1; SMN2TDP1LMNA
SCHEMBL2241896 0.72 RAB9A (1.00) NPC1RAB9ASMN1; SMN2POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed