SCHEMBL20103550

SCHEMBL20103550

CNc1ccc(OCc2nc3ccccc3[nH]2)cc1C

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 11/20 0.64
RAB9A P51151 11/20 0.64
SMN1; SMN2 Q16637 9/20 0.64
TP53 P04637 3/20 0.64
KMT2A Q03164 2/20 0.64
LMNA P02545 2/20 0.64
HTT P42858 2/20 0.64
MEN1 O00255 1/20 0.64
GAA P10253 1/20 0.64
MAPK1 P28482 1/20 0.64
ALDH1A1 P00352 2/20 0.60
TSHR P16473 1/20 0.59
POLB P06746 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
PKM P14618 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5007637 0.79 NPC1 (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL2248644 0.79 NPC1 (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL20103483 0.77 ALOX5 (0.53) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL20103473 0.77 ALOX5 (0.67) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL2246129 0.76 NPC1 (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL15552040 0.76 NPC1 (0.72) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL15063375 0.76 NPC1 (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL2241896 0.75 RAB9A (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A
SCHEMBL9719844 0.75 PDE10A (0.60) CYP1A2
SCHEMBL2245506 0.73 RAB9A (1.00) NPC1RAB9ASMN1; SMN2TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018077898-A1 N,N'-DIARYLUREA, N,N'-DIARYLTHIOUREA AND N,N'-DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE UNIVERSITÄT INNSBRUCK (AT) 2018-05-03 WO disclosed
EP-3315495-A1 N,N' -DIARYLUREA, N,N' -DIARYLTHIOUREA AND N,N' -DIARYLGUANIDINO COMPOUNDS FOR USE IN TREATMENT AND PREVENTION OF INFLAMMATORY DISEASE Universität Innsbruck (AT) 2018-05-02 EP disclosed