SCHEMBL20108429

SCHEMBL20108429

Cc1cc(Cl)c(-c2ccc(C(C)(C)C)cc2)c(C(F)(F)F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
RAPGEF4 Q8WZA2 3/20 0.36
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
PDK2 Q15119 1/20 0.35
FFAR1 O14842 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
GRIA2 P42262 1/20 0.34
GRIA4 P48058 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20108400 0.75 PDK2 (0.33) RAPGEF4PDK2
SCHEMBL5953676 0.74 TSHR (0.52) TSHRAKR1C2AKR1C1KIF11
SCHEMBL25844613 0.74 AR (0.49) AKR1C2FFAR4GABRPGABRDGABRA1
SCHEMBL22031352 0.70 PDK2 (0.48) TSHRRAPGEF4PDK2GABRPGABRD
SCHEMBL1622079 0.69 RXRA (0.47) TSHRAKR1C2AKR1C1KIF11
SCHEMBL3480563 0.69 GABRP (0.53) RAPGEF4GABRPGABRDGABRA1GABRB1
SCHEMBL20108386 0.69 AR (0.45) TSHRRAPGEF4AKR1C2PDK2FFAR4
SCHEMBL18272233 0.69 SMN1; SMN2 (0.40) TSHRRAPGEF4FFAR4
SCHEMBL4792259 0.69 PDE2A (0.51) RAPGEF4GABRA2GABRB2RAPGEF3KIF11
SCHEMBL1104686 0.69 IDO1 (0.44) RAPGEF4RAPGEF3KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964635-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2018-05-02 EP disclosed