SCHEMBL20108400

SCHEMBL20108400

Cc1cc(Cl)c(-c2ccc(C3(C)CCC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.33
HSD11B1 P28845 2/20 0.33
RAPGEF4 Q8WZA2 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
HTT P42858 1/20 0.31
CCR2 P41597 2/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20108429 0.75 TSHR (0.38) PDK2RAPGEF4
SCHEMBL25844613 0.68 AR (0.49)
SCHEMBL24394081 0.66 SLC6A3 (0.49) HSD11B1OPRM1OPRL1
SCHEMBL8297897 0.65 MAOB (0.40) HSD11B1OPRM1OPRK1OPRL1
SCHEMBL13197431 0.64 SLC6A3 (0.51) HSD11B1OPRM1OPRL1
SCHEMBL22031352 0.64 PDK2 (0.48) PDK2HSD11B1RAPGEF4
SCHEMBL22686809 0.64 RAB9A (0.36) HSD11B1HTT
SCHEMBL436499 0.64 SLC6A4 (0.46) HSD11B1CCR2OPRK1
SCHEMBL20108386 0.64 AR (0.45) PDK2HSD11B1RAPGEF4
SCHEMBL18272233 0.63 SMN1; SMN2 (0.40) RAPGEF4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964635-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2018-05-02 EP disclosed