SCHEMBL20108955

SCHEMBL20108955

CCCc1nccc(CI)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.36
KDM4E B2RXH2 4/20 0.35
LMNA P02545 2/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
NOS2 P35228 1/20 0.34
SLC19A2 O60779 1/20 0.34
USP2 O75604 1/20 0.34
CASP1 P29466 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ALDH1A1 P00352 3/20 0.32
HPGD P15428 2/20 0.32
GAA P10253 1/20 0.32
SREBF2 Q12772 7/20 0.31
MAPT P10636 2/20 0.30
NPC1 O15118 1/20 0.30
PKM P14618 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27592765 0.86 KDM4E (0.42) TLR8KDM4ELMNACYP3A4TSHR
Ammonia Solution, Strong SCHEMBL27648732 0.84 KDM4E (0.41) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL16248159 0.84 KDM4E (0.37) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL14424238 0.81 SORD (0.31)
SCHEMBL16815708 0.81 KDM4E (0.39) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL20109822 0.78 LMNA (0.40) LMNANOS2TDP1ALDH1A1L3MBTL1
SCHEMBL14234022 0.77 KCNH2 (0.41) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL15196257 0.76 NOS2 (0.36) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL8176767 0.76 KDM4E (0.37) TLR8KDM4ELMNACYP3A4TSHR
SCHEMBL20109474 0.74 MTNR1A (0.39) KDM4ETDP1HPGDNPC1PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed