SCHEMBL20108966

SCHEMBL20108966

CNC(=O)CCc1nc(CI)ccc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.38
MTNR1B P49286 1/20 0.38
NR4A2 P43354 1/20 0.36
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPK1 P28482 2/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
PCNA P12004 1/20 0.33
POLB P06746 1/20 0.33
TRPV3 Q8NET8 1/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
MPO P05164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015424 0.87 MAPK1 (0.39) MTNR1AMTNR1BNR4A2NPC1TP53
SCHEMBL20108965 0.76 MTNR1A (0.47) MTNR1AMTNR1BNR4A2NPC1TP53
SCHEMBL14234687 0.75 MAPT (0.40) TP53MPOLMNAADORA2AADORA1
SCHEMBL20109474 0.72 MTNR1A (0.39) MTNR1AMTNR1BNR4A2NPC1TP53
SCHEMBL20109473 0.70 MTNR1A (0.39) MTNR1AMTNR1BHDAC1CCNCCDK8
SCHEMBL19287608 0.67 HPGD (0.34) NPC1HDAC1HDAC6RAB9AALDH1A1
SCHEMBL4023871 0.67 DAO (0.41) MTNR1AMTNR1BNR4A2MAPK1HDAC1
SCHEMBL20108967 0.67 HTT (0.39) MTNR1AMTNR1BNR4A2NPC1TP53
SCHEMBL8979538 0.65 TP53 (0.51) MTNR1AMTNR1BNR4A2NPC1TP53
SCHEMBL8027585 0.65 MPO (0.50) MTNR1AMTNR1BCCNCCDK8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed