SCHEMBL20108967

SCHEMBL20108967

CNC(=O)CCc1nc(C)cc(CI)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
HSP90AB1 P08238 1/20 0.37
MAPT P10636 2/20 0.36
MTNR1A P48039 2/20 0.36
MTNR1B P49286 1/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
NR4A2 P43354 1/20 0.34
PCNA P12004 1/20 0.33
POLB P06746 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015430 0.87 HTT (0.40) HTTHSP90AB1MAPTMTNR1AMTNR1B
SCHEMBL20109474 0.77 MTNR1A (0.39) MTNR1AMTNR1BKDM4ENPC1TP53
SCHEMBL20109816 0.74 NOS3 (0.43) HTTKMT2AALDH1A1MEN1
SCHEMBL20108965 0.71 MTNR1A (0.47) MTNR1AMTNR1BNPC1TP53CYP1A2
SCHEMBL16015429 0.69 TP53 (0.36) MTNR1AMTNR1BKDM4ENPC1TP53
SCHEMBL20110098 0.68 HTT (0.54) HTTKMT2AKDM4ETP53CYP1A2
SCHEMBL7457649 0.67 HTT (0.48) HTTMAPTKMT2AKDM4EALDH1A1
SCHEMBL20108966 0.67 MTNR1A (0.38) MTNR1AMTNR1BNPC1TP53CYP1A2
SCHEMBL27326931 0.66 ALPL (0.41) HSP90AB1NPC1TP53CYP1A2CYP2C9
SCHEMBL16015426 0.66 TP53 (0.41) MAPTMTNR1AMTNR1BKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed