SCHEMBL16985359

SCHEMBL16985359

CCOC(=O)C(C)(C)n1ncc(C)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.39
CYP4A11 Q02928 3/20 0.39
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 2/20 0.36
ABCB11 O95342 1/20 0.36
TSHR P16473 1/20 0.36
HTR2A P28223 1/20 0.36
PMP22 Q01453 1/20 0.36
PPARA Q07869 1/20 0.36
PIN1 Q13526 1/20 0.35
CYP2C19 P33261 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
MMP8 P22894 1/20 0.34
CNR2 P34972 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GAA P10253 1/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21850227 0.84 ALDH1A1 (0.39) CYP4F2CYP4A11CYP3A4CYP1A2ABCB11
SCHEMBL18383144 0.79 ALDH1A1 (0.49) ALDH1A1KMT2AMEN1SMN1; SMN2HPGD
SCHEMBL12960396 0.78 CYP1A2 (0.37) CYP3A4CYP1A2TSHRCYP2C19ALDH1A1
SCHEMBL16985342 0.77 GRIA1 (0.37) ALDH1A1KMT2AMEN1KDM4EGRIA1
SCHEMBL30867737 0.76 PDE4A (0.35) CYP4F2CYP4A11CYP3A4CYP1A2ABCB11
SCHEMBL16985341 0.75 GRIA1 (0.36) KMT2AGRIA1GRIA2GRIA3GRIA4
SCHEMBL574545 0.73 RAB9A (0.48) CYP3A4TSHRCYP2C19ALDH1A1KMT2A
SCHEMBL9877609 0.73 SMN1; SMN2 (0.51) CYP3A4CYP1A2TSHRCYP2C19ALDH1A1
SCHEMBL15339562 0.72 ALDH1A1 (0.38) CYP4F2CYP4A11ALDH1A1KMT2AMEN1
SCHEMBL20117304 0.72 KMO (0.48) CYP4F2CYP4A11CYP1A2TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015113452-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2015-08-06 WO disclosed