SCHEMBL20124669

SCHEMBL20124669

C=COCCCc1ccc(Cc2cc(Br)ccc2C)cc1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
SLC5A1 P13866 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
SLC5A2 P31639 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20124703 0.92 TAAR1 (0.33) TAAR1PDE3BPDE3A
SCHEMBL499758 0.84 HTR2A (0.32) CNR1CNR2GPR55SLC5A1LMNA
SCHEMBL500101 0.76 HTR2A (0.33) SLC5A1LMNASLC5A2
SCHEMBL1010022 0.73 ALDH1A1 (0.44) SLC5A1TAAR1LMNASLC5A2PDE3B
SCHEMBL15748708 0.72 PKM (0.47) SLC5A1KDM4ELMNASLC5A2
SCHEMBL37695 0.72 KDM4E (0.44) SLC5A1KDM4ESLC5A2PDE3BPDE3A
SCHEMBL180996 0.71 SLC5A1 (0.46) CNR2SLC5A1LMNASLC5A2
SCHEMBL17175 0.70 ESR1 (0.45) KDM4E
SCHEMBL15741057 0.70 CCR5 (0.47) SLC5A1
SCHEMBL2810557 0.70 KDM4E (0.41) TAAR1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3318562-A2 BENZYLBENZENE DERIVATIVES AND METHODS OF USE Theracos Sub, LLC (US) 2018-05-09 EP disclosed