SCHEMBL20125018

SCHEMBL20125018

CNCc1cc(C)cnc1N

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.50
NOS2 P35228 2/20 0.50
NOS1 P29475 1/20 0.50
CYP2A6 P11509 2/20 0.37
SLC6A4 P31645 10/20 0.36
SLC6A2 P23975 9/20 0.36
SLC6A3 Q01959 7/20 0.36
CYP2D6 P10635 1/20 0.34
KCNH2 Q12809 1/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093855 0.79 KMT2A (0.48) SLC6A4SLC6A2KCNH2LMNA
SCHEMBL31587245 0.78 NOS3 (0.56) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL12647715 0.78 NOS3 (0.56) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL13283349 0.78 NOS3 (0.56) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL22945605 0.77 SLC6A2 (0.36) SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL15828598 0.77 DHFR (0.33) NOS3NOS2NOS1SLC6A4SLC6A2
SCHEMBL20465810 0.76 NOS3 (0.54) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL17480023 0.76 NOS3 (0.54) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL20465809 0.74 LMNA (0.55) NOS3NOS2NOS1CYP2A6LMNA
SCHEMBL20124986 0.73 NOS3 (0.50) NOS3NOS2NOS1CYP2A6SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190077762-A1 QUINOLONE COMPOUND OTSUKA PHARMA CO LTD (JP) 2019-03-14 US disclosed
EP-3318557-A2 QUINOLONE COMPOUND Otsuka Pharmaceutical Co., Ltd. (JP) 2018-05-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077762-A1 QUINOLONE COMPOUND HAX1, NQO2, NHERF1 NOS3 2969/4885NOS2 3433/4885NOS1 2630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.