SCHEMBL2013138

SCHEMBL2013138

C[C@H]1CN(Cc2ccn(-c3cccnc3N3CCC(Oc4ccc(F)cc4)CC3)n2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLNR O43193 7/20 0.65
MGLL Q99685 1/20 0.41
CXCR3 P49682 3/20 0.37
PDK1 Q15118 1/20 0.37
PDK2 Q15119 1/20 0.37
PDK3 Q15120 1/20 0.37
PDK4 Q16654 1/20 0.37
CCR1 P32246 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC3 O15379 1/20 0.36
CYP2C9 P11712 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
MAPKAPK3 Q16644 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
CHRM4 P08173 1/20 0.36
ACACB O00763 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010301 0.93 MLNR (0.66) MLNRMGLLCXCR3PDK1PDK2
SCHEMBL3138321 0.90 MLNR (0.72) MLNRMGLLCCR1ALDH1A1KMT2A
SCHEMBL3134434 0.83 MLNR (0.73) MLNRMGLL
SCHEMBL2007837 0.81 MLNR (0.73) MLNRALDH1A1KMT2A
SCHEMBL2013140 0.81 MLNR (0.61) MLNRALDH1A1KMT2A
SCHEMBL3128327 0.79 MLNR (0.85) MLNRCHRM4
SCHEMBL2012437 0.72 MLNR (1.00) MLNR
SCHEMBL2010214 0.71 MLNR (0.46) MLNRPDK1PDK2PDK3PDK4
SCHEMBL2008090 0.70 MLNR (0.73) MLNR
SCHEMBL2010191 0.69 PDK1 (0.50) MGLLPDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7964602-B2 Biaryl compounds useful as agonists of the Gpr38 receptor GLAXO GROUP LIMITED (GB) 2011-06-21 US disclosed