SCHEMBL20134858

SCHEMBL20134858

Cc1ccc(C(=O)C2CCN(C(=O)OC(C)(C)C)CC2)nc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.55
GPR119 Q8TDV5 8/20 0.53
HPGD P15428 1/20 0.50
PTPN2 P17706 1/20 0.50
PTPN1 P18031 1/20 0.50
PTPN6 P29350 1/20 0.50
RECQL P46063 1/20 0.48
STS P08842 4/20 0.47
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17827895 0.93 KMT2A (0.50) KMT2AGPR119HPGDPTPN2PTPN1
SCHEMBL17827899 0.88 GPR119 (0.43) KMT2AGPR119HPGD
SCHEMBL12919132 0.87 PTPN2 (0.49) KMT2AGPR119HPGDPTPN2PTPN1
SCHEMBL20135438 0.86 KMT2A (0.54) KMT2AGPR119HPGDPTPN2PTPN1
SCHEMBL12367647 0.84 RECQL (0.48) KMT2AGPR119HPGDPTPN2PTPN1
SCHEMBL17820470 0.82 TDP1 (0.57) KMT2AGPR119
SCHEMBL406827 0.81 GPR119 (0.62) GPR119HPGDPTPN2PTPN1PTPN6
SCHEMBL14113587 0.81 KMT2A (0.71) KMT2AGPR119HPGDPTPN2PTPN1
SCHEMBL390649 0.80 USP30 (0.48) GPR119HPGDPTPN2PTPN1PTPN6
SCHEMBL17819837 0.79 KDM4A (0.47) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10407408-B2 Imide derivatives and use thereof as medicine MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-09-10 US disclosed
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MITSUBISHI TANABE PHARMA CORPORATION (JP) 2019-03-14 US disclosed
EP-3321256-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE Mitsubishi Tanabe Pharma Corporation (JP) 2018-05-16 EP disclosed
CN-107922347-A New imide derivative and its purposes as medicine 田边三菱制药株式会社 2018-04-17 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077787-A1 NOVEL IMIDE DERIVATIVES AND USE THEREOF AS MEDICINE MMP9, MMP10, MMP1 KMT2A 2568/4885GPR119 799/4885HPGD 74/4885
US-10407408-B2 Imide derivatives and use thereof as medicine MMP9, MMP2, MMP1 KMT2A 2539/4885GPR119 997/4885HPGD 75/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.