SCHEMBL20139218

SCHEMBL20139218

COC(=O)c1cc(C=O)cn1CC(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
HDAC8 Q9BY41 2/20 0.38
LDHA P00338 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
NR4A2 P43354 1/20 0.31
HTR3A P46098 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C19 P33261 2/20 0.31
HSP90AA1 P07900 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
BRD4 O60885 1/20 0.31
NOTUM Q6P988 2/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16320824 0.85 ALDH1A1 (0.42) ALDH1A1HDAC8CA12CA1CA2
SCHEMBL30838204 0.82 BRD4 (0.39) ALDH1A1HDAC8NR4A2HTR3ASMN1; SMN2
SCHEMBL20139328 0.82 HDAC8 (0.32) ALDH1A1HDAC8
SCHEMBL10565454 0.77 ALDH1A1 (0.38) ALDH1A1HDAC8SMN1; SMN2CYP1A2CYP2C19
SCHEMBL4301396 0.74 KMT2A (0.43) ALDH1A1MAPTKDM4EPOLB
SCHEMBL3387788 0.73 HDAC8 (0.51) ALDH1A1HDAC8NR4A2CYP1A2CYP2C19
SCHEMBL4305907 0.73 LMNA (0.38) ALDH1A1HDAC8LDHAMAPTNOTUM
SCHEMBL24435291 0.73 MAPK10 (0.52) ALDH1A1HDAC8MAPTBRD4KDM4E
SCHEMBL4308531 0.71 LMNA (0.43) ALDH1A1CYP1A2CYP2C19MAPTHPGD
SCHEMBL4306412 0.71 KMT2A (0.42) ALDH1A1HDAC8SMN1; SMN2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed