SCHEMBL4305907

SCHEMBL4305907

COC(=O)c1cc(C=O)cn1CC(=O)c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
P4HB P07237 1/20 0.37
NOTUM Q6P988 1/20 0.37
TAS1R3 Q7RTX0 2/20 0.36
TAS1R1 Q7RTX1 2/20 0.36
TAS1R2 Q8TE23 2/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TP53 P04637 1/20 0.36
RXRA P19793 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36
ERN1 O75460 2/20 0.35
LDHA P00338 1/20 0.35
HDAC8 Q9BY41 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8020013 0.88 GRIN2B (0.39) LMNATAS1R3TAS1R1TAS1R2MAPT
SCHEMBL4311981 0.85 LMNA (0.44) LMNATAS1R3TAS1R1TAS1R2MAPT
SCHEMBL4301396 0.82 KMT2A (0.43) TAS1R3TAS1R1MAPTALDH1A1KDM4E
SCHEMBL4306412 0.81 KMT2A (0.42) LMNAMAPTALDH1A1GRIN2BERN1
SCHEMBL4308531 0.78 LMNA (0.43) LMNAMAPTALDH1A1KDM4E
SCHEMBL4306380 0.78 CYP1A2 (0.43) LMNAMAPTALDH1A1TP53KDM4E
SCHEMBL4302800 0.76 CDYL2 (0.49) LMNAMAPTALDH1A1TP53KDM4E
SCHEMBL20139218 0.73 ALDH1A1 (0.38) NOTUMMAPTALDH1A1LDHAHDAC8
SCHEMBL16320824 0.73 ALDH1A1 (0.42) LMNAMAPTALDH1A1HDAC8KDM4E
SCHEMBL14012580 0.72 NOTUM (0.64) LMNAP4HBNOTUMTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed