SCHEMBL20139604

SCHEMBL20139604

O=C[C@H](c1cccnn1)c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.40
SLC6A9 P48067 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
MAPKAPK2 P49137 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5071497 0.81 NFE2L2 (0.38) HDAC4CES2CES1
SCHEMBL20139709 0.81 HDAC4 (0.38) HDAC4SLC6A9
SCHEMBL9347326 0.77 CES2 (0.42) CES2CES1
SCHEMBL20139617 0.74 HDAC4 (0.41) HDAC4CES2CES1MAPKAPK2
SCHEMBL17316873 0.73 HDAC4 (0.49) HDAC4SLC6A9CES2CES1
SCHEMBL20141623 0.72 HDAC4 (0.37) HDAC4SLC6A9
SCHEMBL1515751 0.71 IDO1 (0.46) CES2CES1
SCHEMBL14743495 0.68 CES2 (0.36) HDAC4CES2CES1
SCHEMBL2724490 0.68 CES2 (0.36) CES2CES1
SCHEMBL9363514 0.68 IDO1 (0.36) HDAC4CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed