SCHEMBL20139617

SCHEMBL20139617

O=C[C@H](c1cnccn1)c1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 6/20 0.41
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPKAPK2 P49137 1/20 0.32
ROCK2 O75116 1/20 0.32
NFE2L2 Q16236 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
GAA P10253 1/20 0.30
PIM1 P11309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5071497 0.83 NFE2L2 (0.38) HDAC4NFE2L2CES2CES1
SCHEMBL20139680 0.81 HDAC4 (0.39) HDAC4HPGDHSD17B10ROCK2
SCHEMBL1515803 0.78 SLC6A2 (0.39) HPGDGAA
SCHEMBL9347326 0.76 CES2 (0.42) NFE2L2CES2CES1GAA
SCHEMBL20139604 0.74 HDAC4 (0.40) HDAC4MAPKAPK2CES2CES1
SCHEMBL20139663 0.73 ROCK2 (0.39) HDAC4HPGDHSD17B10ROCK2ALOX5AP
SCHEMBL15109715 0.70 HDAC4 (0.39) HDAC4NFE2L2CES2CES1
SCHEMBL1515751 0.70 IDO1 (0.46) CES2CES1GAA
SCHEMBL5739585 0.69 HDAC4 (0.34) HDAC4HPGDHSD17B10CES2CES1
SCHEMBL14743495 0.67 CES2 (0.36) HDAC4NFE2L2CES2CES1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed