SCHEMBL20141623

SCHEMBL20141623

NC[C@@H](c1cccnn1)c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.37
IDO1 P14902 2/20 0.35
TDO2 P48775 2/20 0.35
SLC6A9 P48067 1/20 0.34
ROCK2 O75116 1/20 0.34
CNR2 P34972 1/20 0.34
TAAR1 Q96RJ0 2/20 0.33
HTR2A P28223 1/20 0.33
CYP1A2 P05177 1/20 0.33
F2 P00734 1/20 0.32
CYP19A1 P11511 1/20 0.32
GAA P10253 1/20 0.32
GOT1 P17174 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3712034 0.78 HTR2A (0.54) SLC6A9TAAR1HTR2ACYP1A2SLC6A2
SCHEMBL20139663 0.77 ROCK2 (0.39) HDAC4IDO1TDO2ROCK2TAAR1
SCHEMBL17316873 0.73 HDAC4 (0.49) HDAC4SLC6A9CYP1A2GAA
SCHEMBL3910983 0.72 TAAR1 (0.60) IDO1TDO2TAAR1HTR2ACYP1A2
SCHEMBL20139604 0.72 HDAC4 (0.40) HDAC4SLC6A9
SCHEMBL7297048 0.70 SLC6A2 (0.42) IDO1TDO2HTR2ACYP2D6SLC6A2
SCHEMBL20161464 0.69 TAAR1 (0.38) IDO1TAAR1CYP1A2CYP19A1GOT1
SCHEMBL20139709 0.69 HDAC4 (0.38) HDAC4SLC6A9
SCHEMBL27490477 0.69 CYP1A2 (0.40) CYP1A2GOT1
SCHEMBL6001389 0.68 HRH1 (0.54) IDO1TDO2CNR2TAAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed