SCHEMBL20139663

SCHEMBL20139663

NC[C@@H](c1cnccn1)c1ccccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.39
HDAC4 P56524 1/20 0.38
CYP19A1 P11511 1/20 0.36
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
HPGD P15428 2/20 0.33
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
HTR2A P28223 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
TERT O14746 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141623 0.77 HDAC4 (0.37) ROCK2HDAC4CYP19A1IDO1TDO2
SCHEMBL7297048 0.75 SLC6A2 (0.42) IDO1TDO2CYP2D6HRH1ALDH1A1
SCHEMBL20139617 0.73 HDAC4 (0.41) ROCK2HDAC4HPGDHSD17B10ALOX5AP
SCHEMBL6203371 0.73 SMN1; SMN2 (0.40) HDAC4ALDH1A1FEN1
SCHEMBL3910983 0.71 TAAR1 (0.60) CYP19A1IDO1TDO2CYP2D6HRH1
SCHEMBL20161327 0.70 NPC1 (0.38) CYP19A1IDO1LOXL2CYP2D6TAAR1
SCHEMBL20773226 0.70 CTSA (0.44) IDO1TDO2TAAR1
SCHEMBL20139680 0.70 HDAC4 (0.39) ROCK2HDAC4HPGDKMT2AHSD17B10
SCHEMBL5739585 0.69 HDAC4 (0.34) HDAC4HPGDHSD17B10GAA
SCHEMBL7521138 0.68 SLC6A2 (0.43) CYP2D6HRH1ALDH1A1HTR2ATAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed