SCHEMBL20139680

SCHEMBL20139680

ON=C[C@H](c1cnccn1)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.39
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KMT2A Q03164 1/20 0.30
ROCK2 O75116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139617 0.81 HDAC4 (0.41) HDAC4HPGDHSD17B10ROCK2
SCHEMBL20139709 0.76 HDAC4 (0.38) HDAC4
SCHEMBL21229255 0.74 MAPK9 (0.37) KMT2A
SCHEMBL20139663 0.70 ROCK2 (0.39) HDAC4HPGDHSD17B10KMT2AROCK2
SCHEMBL5739585 0.66 HDAC4 (0.34) HDAC4HPGDHSD17B10
SCHEMBL5071497 0.64 NFE2L2 (0.38) HDAC4KMT2A
SCHEMBL20161327 0.64 NPC1 (0.38)
SCHEMBL11215460 0.62 SLC6A2 (0.52)
SCHEMBL11215459 0.62 SLC6A2 (0.52)
SCHEMBL1515803 0.62 SLC6A2 (0.39) HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538520-A2 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2019-09-18 EP disclosed
WO-2018089330-A2 SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed