SCHEMBL20139745

SCHEMBL20139745

CC(C)(C)C1(C)CN(c2cccc3cc[nH]c23)CCN1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.37
PDPK1 O15530 1/20 0.34
BCHE P06276 4/20 0.34
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
AR P10275 1/20 0.32
IDO1 P14902 1/20 0.32
PTPN11 Q06124 1/20 0.31
HASPIN Q8TF76 1/20 0.31
BACE1 P56817 1/20 0.31
GOT1 P17174 2/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
RBP4 P02753 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20141537 0.74 KEAP1 (0.47) KEAP1PDPK1BCHEGOT1GAA
SCHEMBL20142570 0.72 KEAP1 (0.38) KEAP1PDPK1BCHENR3C1PGR
SCHEMBL30885785 0.71 IDO1 (0.48) BCHEIDO1BACE1MAPT
SCHEMBL5205461 0.71 IDO1 (0.48) BCHEIDO1BACE1MAPT
SCHEMBL20140928 0.70 SLC6A7 (0.42) GAAMAPT
SCHEMBL20142085 0.69 KLKB1 (0.30)
SCHEMBL25267550 0.68 MEN1 (0.36) KEAP1IDO1PTPN11GAAMAPT
SCHEMBL3296720 0.68 GOT1 (0.42) KEAP1PDPK1BCHEGOT1GAA
SCHEMBL3624025 0.67 AR (0.51) ARGAAMAPT
Trifluoroacetic Acid SCHEMBL30839779 0.67 BACE1 (0.46) KEAP1BACE1HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed