SCHEMBL20140448

SCHEMBL20140448

CC(C)(C)C(CNC(=O)O)n1ncc(-c2ccccc2)c1CCl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
LPAR1 Q92633 2/20 0.33
NPC1 O15118 2/20 0.33
NFKB1 P19838 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
MAPT P10636 2/20 0.33
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
CNR2 P34972 1/20 0.32
GPR119 Q8TDV5 3/20 0.32
SHMT1 P34896 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140431 0.91 SMN1; SMN2 (0.36) PTGIRSMN1; SMN2KDM5AKDM4CKDM5B
SCHEMBL20140105 0.67 CKS1B (0.44) PTGIRSMN1; SMN2KDM4EALDH1A1HPGD
SCHEMBL20140446 0.65 PTGIR (0.44) PTGIRSMN1; SMN2LPAR1NPC1NFKB1
SCHEMBL20140432 0.61 CKS1B (0.45) PTGIRSMN1; SMN2DRD2
SCHEMBL21247485 0.60 CNR1 (0.43) SMN1; SMN2NPC1RAB9AMAPTCNR2
SCHEMBL27996913 0.60 PTGIR (0.49) PTGIRSMN1; SMN2LPAR1NPC1NFKB1
SCHEMBL9877332 0.59 MAPT (0.54) PTGIRSMN1; SMN2NPC1NFKB1RAB9A
SCHEMBL20140430 0.59 PTGIR (0.43) PTGIRSMN1; SMN2LPAR1NPC1NFKB1
SCHEMBL11491087 0.59 PTGIR (0.79) PTGIRSMN1; SMN2KDM4EHSD17B10
SCHEMBL25731618 0.58 CYP11B2 (0.47) PTGIRSMN1; SMN2LPAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed