SCHEMBL20145024

SCHEMBL20145024

CN1CCCC(Oc2ccc(F)cn2)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.48
IL1B P01584 1/20 0.45
NLRP3 Q96P20 1/20 0.45
CHRM1 P11229 3/20 0.44
CHRM3 P20309 3/20 0.44
CHRM2 P08172 2/20 0.44
CHRM5 P08912 2/20 0.44
CHRM4 P08173 1/20 0.44
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
TLR7 Q9NYK1 2/20 0.39
HRH3 Q9Y5N1 2/20 0.39
ATM Q13315 1/20 0.39
ATR Q13535 1/20 0.39
NTMT1 Q9BV86 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19865665 0.93 TDO2 (0.54) TDO2CHRM1CHRM3CHRM2CHRM5
SCHEMBL19865633 0.93 TDO2 (0.54) TDO2CHRM1CHRM3CHRM2CHRM5
SCHEMBL20069366 0.93 TDO2 (0.54) TDO2CHRM1CHRM3CHRM2CHRM5
SCHEMBL20147962 0.85 TDO2 (0.61) TDO2TLR7HRH3
SCHEMBL16382664 0.85 TDO2 (0.45) TDO2TLR7
SCHEMBL1926965 0.83 IL1B (0.43) TDO2IL1BNLRP3CHRM1CHRM3
SCHEMBL20145059 0.83 L3MBTL1 (0.49) IL1BNLRP3CHRM1CHRM3CHRM2
SCHEMBL20144750 0.83 IL1B (0.55) IL1BNLRP3
SCHEMBL20145221 0.83 IL1B (0.55) IL1BNLRP3
SCHEMBL19641554 0.80 TDO2 (0.45) TDO2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed