SCHEMBL20149228

SCHEMBL20149228

CCc1c(F)cc(N)cc1F

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
USP7 Q93009 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21736856 0.86 NOS3 (0.35) TAAR1ALDH1A1TSHRNOS3NOS2
SCHEMBL10228073 0.84 CYP3A4 (0.41) TAAR1ALDH1A1TSHR
SCHEMBL12184907 0.80 TAAR1 (0.42) TAAR1ALDH1A1TSHRNOS3NOS2
SCHEMBL20076496 0.78 TBK1 (0.30)
SCHEMBL1547845 0.78 RIPK1 (0.40) TAAR1ALDH1A1
SCHEMBL5522542 0.78 TAAR1 (0.37) TAAR1ALDH1A1TSHR
SCHEMBL9336 0.76 SELL (0.33) TAAR1ALDH1A1TSHRNOS3NOS2
SCHEMBL29467951 0.76 TAAR1 (0.41) TAAR1ALDH1A1TSHR
SCHEMBL15247375 0.76 PTGS2 (0.36) TAAR1
SCHEMBL9494017 0.75 TAAR1 (0.33) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11834440-B2 Beta-lactam derivatives for the treatment of diseases INSILICO MEDICINE IP LIMITED (HK) 2023-12-05 US disclosed
EP-3611165-B1 PYRIDONE COMPOUND, AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE HAVING THIS AS ACTIVE COMPONENT MITSUI CHEMICALS CROP & LIFE SOLUTIONS INC (JP) 2023-08-16 EP disclosed
EP-3611165-A1 PYRIDONE COMPOUND, AND AGRICULTURAL AND HORTICULTURAL FUNGICIDE HAVING THIS AS ACTIVE COMPONENT Mitsui Chemicals Agro, Inc. (JP) 2020-02-19 EP disclosed
WO-2018089373-A9 STEROIDS AND PROTEIN-CONJUGATES THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2018-07-12 WO disclosed
WO-2018089373-A2 STEROIDS AND PROTEIN-CONJUGATES THEREOF REGENERON PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11834440-B2 Beta-lactam derivatives for the treatment of diseases QPCT, QPCTL, BCAT1 TAAR1 4364/4885ALDH1A1 2194/4885TSHR 3851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.