SCHEMBL20155016

SCHEMBL20155016

CN(C)CCn1cc2c(Cl)nccc2n1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.38
FERMT2 Q96AC1 1/20 0.36
PDE4D Q08499 1/20 0.34
HTR6 P50406 5/20 0.34
ADRA1A P35348 1/20 0.34
HRH1 P35367 1/20 0.34
ADRA1B P35368 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.34
TGFBR1 P36897 4/20 0.33
HRH3 Q9Y5N1 2/20 0.33
KDM5A P29375 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
MAP4K4 O95819 2/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR7 P34969 1/20 0.32
IRAK1 P51617 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23531689 0.81 PDE4D (0.43) PDE4D
SCHEMBL20155347 0.80 MAT2A (0.38) PDE4D
SCHEMBL20155042 0.79 MAP4K4 (0.42) PDE4DIRAK4MAP4K4
SCHEMBL17873844 0.74 ADORA2A (0.40)
SCHEMBL20155108 0.73 TGFBR1 (0.45) TGFBR1HTR2C
SCHEMBL12913813 0.71 KMT2A (0.40) KDM5AKDM5B
SCHEMBL22216456 0.70 ALDH1A1 (0.44) CNR2
SCHEMBL20155563 0.70 CNR2 (0.42) CNR2PDE4DHTR6KDM5B
SCHEMBL25239263 0.70 DGAT1 (0.33) PDE4D
SCHEMBL17221286 0.68 GAA (0.52) TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed