SCHEMBL20155042

SCHEMBL20155042

COCCn1cc2c(Cl)nccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.42
EGFR P00533 1/20 0.42
FRK P42685 1/20 0.42
MAPK9 P45984 1/20 0.42
CSNK1D P48730 1/20 0.42
SLK Q9H2G2 1/20 0.42
LRRK2 Q5S007 2/20 0.40
MPO P05164 2/20 0.38
PTPN11 Q06124 1/20 0.38
PDE4D Q08499 3/20 0.37
IRAK4 Q9NWZ3 3/20 0.33
PDE4B Q07343 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DYRK1A Q13627 2/20 0.32
NFATC1 O95644 1/20 0.32
GSK3B P49841 1/20 0.32
ATM Q13315 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155044 0.82 MPO (0.38) MAP4K4EGFRFRKMAPK9CSNK1D
SCHEMBL23531689 0.81 PDE4D (0.43) LRRK2MPOPDE4DPDE4BKDM4E
SCHEMBL20155347 0.80 MAT2A (0.38) PTPN11PDE4DPDE4BSMN1; SMN2KDM4E
SCHEMBL20155016 0.79 CNR2 (0.38) MAP4K4PDE4DIRAK4
SCHEMBL22216456 0.76 ALDH1A1 (0.44) SMN1; SMN2KDM4EALDH1A1GSK3B
SCHEMBL21631825 0.75 PTPN11 (0.41) MAP4K4EGFRFRKMAPK9CSNK1D
SCHEMBL25239263 0.75 DGAT1 (0.33) PDE4D
SCHEMBL23386491 0.75 KDR (0.43) MAP4K4EGFRFRKMAPK9CSNK1D
SCHEMBL17873844 0.74 ADORA2A (0.40) CSNK1DPTPN11SMN1; SMN2KDM4EALDH1A1
SCHEMBL20155060 0.73 F2RL3 (0.33) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115806551-A Pyrazole-containing polycyclic derivative, pharmaceutically acceptable salt thereof, and preparation method and application thereof 优领医药科技(香港)有限公司 2023-03-17 CN disclosed
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed