SCHEMBL20155093

SCHEMBL20155093

CC(C)n1cc2c(Br)cn(C)c(=O)c2n1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 1/20 0.36
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
BRD4 O60885 2/20 0.32
BRD2 P25440 2/20 0.32
BRD3 Q15059 2/20 0.32
CREBBP Q92793 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155332 0.89 ADORA2A (0.36) MAT2AADORA2AADORA1BRD4BRD2
SCHEMBL20155066 0.80 MAT2A (0.34) MAT2AADORA2AADORA1BRD4
SCHEMBL20154927 0.74 MAT2A (0.40) MAT2A
SCHEMBL20155133 0.68 ADORA2A (0.37) ADORA2A
SCHEMBL20155003 0.67 BRD4 (0.36) MAT2AADORA2AADORA1BRD4
SCHEMBL20155089 0.66 PSMB5 (0.31) BRD4
SCHEMBL19869860 0.66 BRD4 (0.49) BRD4
SCHEMBL20155331 0.66 ADORA2A (0.36) MAT2AADORA2AADORA1
SCHEMBL25102855 0.65 KDM4E (0.38) ADORA2AADORA1BRD4
SCHEMBL21224338 0.65 BRD4 (0.36) BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed