SCHEMBL20155367

SCHEMBL20155367

CC(C)n1ncc2c(=O)n(C)cc(Br)c21

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 5/20 0.34
BRD4 O60885 4/20 0.34
BRD2 P25440 2/20 0.34
BRD3 Q15059 2/20 0.34
PDE1C Q14123 2/20 0.34
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 2/20 0.31
PDE9A O76083 1/20 0.31
PDE1A P54750 1/20 0.31
PDE1B Q01064 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
AURKA O14965 1/20 0.30
CDK1 P06493 1/20 0.30
AURKB Q96GD4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28520363 0.80 HTT (0.38) CREBBPBRD4ALDH1A1SMN1; SMN2
SCHEMBL20155328 0.70 HTT (0.41) BRD4KDM4EALDH1A1SMN1; SMN2
SCHEMBL20155369 0.68 KDM4E (0.33) KDM4E
SCHEMBL20155332 0.68 ADORA2A (0.36) CREBBPBRD4BRD2BRD3
SCHEMBL9726416 0.67 ALDH1A1 (0.46) PDE1CKDM4EALDH1A1CYP1A2CYP2C19
SCHEMBL21224811 0.67 BRD4 (0.37) BRD4
SCHEMBL20154923 0.66 BRD4 (0.38) BRD4
SCHEMBL21363594 0.66 IMPDH2 (0.36) PDE1CKDM4EALDH1A1
SCHEMBL30975384 0.66 LMNA (0.35) BRD4ALDH1A1
SCHEMBL16651029 0.65 BRD9 (0.45) BRD4CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed