SCHEMBL20155498

SCHEMBL20155498

CC1(C)OB(c2cc(N)c(Cl)cc2Nc2ccc(F)cc2F)OC1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34
EGFR P00533 2/20 0.34
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
SOS1 Q07889 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
HDAC3 O15379 1/20 0.30
NCOR1 O75376 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155541 0.89 ALDH1A1 (0.40) ALDH1A1LPLLIPGCYP2D6CYP2C19
SCHEMBL20155117 0.83 ALDH1A1 (0.39) ALDH1A1LPLLIPGEGFRCYP2D6
SCHEMBL20155461 0.79 TDO2 (0.38) ALDH1A1LPLLIPGEGFRCA1
SCHEMBL20155588 0.78 ALDH1A1 (0.37) ALDH1A1LPLLIPGEGFRCYP2D6
SCHEMBL25277938 0.76 GAA (0.35) LPLLIPGEGFRGAA
SCHEMBL20155620 0.76 EGFR (0.37) EGFRCA1CA2CA9KMT2A
SCHEMBL21190843 0.74 BRD4 (0.45) ALDH1A1SOS1CA1CA2CA9
SCHEMBL21067071 0.73 GAA (0.35) LPLLIPGEGFRGAA
SCHEMBL20155496 0.72 SOS1 (0.42) ALDH1A1CYP2D6CYP2C19SOS1MAPK13
SCHEMBL772615 0.71 LPL (0.49) ALDH1A1LPLLIPGCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed